Synonyms: 4-(N-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-(trifluoromethoxy)benzyl)sulfamoyl)benzoic acid; 4-[[[3-Chloro-5-(trifluoromethyl)-2-pyridinyl][[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]-benzoic acid
Molecular Formula: C21H13ClF6N2O5S
Molecular Weight: 554.85
Linear Structural Formula: C21H13ClF6N2O5S
MDL Number: MFCD29049510
Purity: >=98% (HPLC)
Storage: 2-8C
Biochem Physiol Actions: RQ-00203078 is an orally available potent and selective TRPM8 antagonist that potently reduces cation currents induced by menthol and other TRPM8 agonists. RQ-00203078 inhibits HSC3 and HSC4 oral squamous carcinoma cell migration and invasion in vitro.